SCHEMBL4697074

SCHEMBL4697074

O=C(O)C1c2sccc2C(NOCc2ccccc2)CN1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
EPHX2 P34913 2/20 0.33
GRIN2B Q13224 1/20 0.33
AGTR2 P50052 3/20 0.33
S1PR5 Q9H228 1/20 0.33
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSK P43235 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
SLC6A1 P30531 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138221 0.90 GPR183 (0.35) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL5254943 0.83 NPC1 (0.38) NPC1RAB9AEPHX2S1PR5SMN1; SMN2
SCHEMBL5255317 0.82 HHAT (0.33)
SCHEMBL5255311 0.82 HHAT (0.33)
SCHEMBL4696597 0.76 NPC1 (0.35) NPC1RAB9AEPHX2GRIN2BSMN1; SMN2
SCHEMBL5187275 0.76 GPR183 (0.39) NPC1RAB9AALDH1A1
SCHEMBL3305431 0.75 LMNA (0.34) NPC1RAB9AEPHX2S1PR5SMN1; SMN2
SCHEMBL4695600 0.74 KEAP1 (0.40) NPC1RAB9A
SCHEMBL5185290 0.73 HHAT (0.34)
SCHEMBL4696326 0.73 AGTR2 (0.33) AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed