SCHEMBL4693843

SCHEMBL4693843

O=C(O)C1NCC(NOCc2ccccc2)c2cnn(-c3ccccc3)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.36
SLC9A1 P19634 1/20 0.35
SLC9A2 Q9UBY0 1/20 0.35
MAPK14 Q16539 1/20 0.35
KHK P50053 1/20 0.35
HPGD P15428 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALPL P05186 1/20 0.34
ALPI P09923 1/20 0.34
ALPG P10696 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4145877 0.90 HTT (0.39) KEAP1NFE2L2LMNAHTTKMT2A
SCHEMBL4695600 0.80 KEAP1 (0.40) KEAP1NFE2L2LMNAHTTKMT2A
SCHEMBL5330841 0.79 TSHR (0.40) NPC1ALDH1A1TSHRRAB9A
SCHEMBL20558125 0.79 ACHE (0.34) LMNANPC1HPGDALDH1A1RAB9A
SCHEMBL4694770 0.76 NPC1 (0.35) NPC1ALDH1A1RAB9A
SCHEMBL4138926 0.75 KEAP1 (0.38) KEAP1NFE2L2LMNAHTTKMT2A
SCHEMBL4696597 0.73 NPC1 (0.35) NPC1ALDH1A1RAB9A
SCHEMBL5187221 0.71 NPC1 (0.37) NPC1HPGDALDH1A1TSHRRAB9A
SCHEMBL20558166 0.71
SCHEMBL20557971 0.70 CCNB2 (0.35) NPC1ALDH1A1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed