SCHEMBL4696655

SCHEMBL4696655

CC1(C)Cc2c(sc(NC(=O)C(c3ccccc3)(c3ccccc3)c3ccccc3)c2C#N)CO1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.63
RAB9A P51151 6/20 0.63
SMN1; SMN2 Q16637 6/20 0.63
ALDH1A1 P00352 6/20 0.63
TP53 P04637 1/20 0.63
KMT2A Q03164 7/20 0.62
MEN1 O00255 6/20 0.62
KDM4E B2RXH2 2/20 0.60
HPGD P15428 2/20 0.52
MAPT P10636 4/20 0.51
EPHB4 P54760 1/20 0.48
RAB7A P51149 4/20 0.48
PLA2G1B P04054 1/20 0.46
GAA P10253 1/20 0.46
CDC42 P60953 1/20 0.46
RAB2A P61019 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CFTR P13569 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15281315 0.78 ALDH1A1 (1.00) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL21247198 0.68 ALDH1A1 (1.00) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL8288608 0.65 KMT2A (0.71) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL15832859 0.65 RAB7A (1.00) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL21260779 0.63 ALDH1A1 (0.66) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL15272485 0.61 KDM4E (0.72) SMN1; SMN2ALDH1A1KMT2AMEN1KDM4E
SCHEMBL14825265 0.61 CFTR (0.80) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL2643514 0.61 ALDH1A1 (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL618553 0.60 ALDH1A1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL2643860 0.60 GCGR (0.49) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620425-B1 SUBSTITUTED 3-CYANOTHIOPHENE ACETAMIDES AS GLUCAGON RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-12-24 EP claimed