SCHEMBL4696826

SCHEMBL4696826

Cc1ccc(C(=O)O)c(C#N)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
KMT2A Q03164 1/20 0.42
SELL P14151 1/20 0.39
SELP P16109 1/20 0.39
MCL1 Q07820 1/20 0.39
HAAO P46952 1/20 0.38
NOTUM Q6P988 2/20 0.38
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
GLO1 Q04760 1/20 0.37
HMGB1 P09429 1/20 0.37
CXCL12 P48061 1/20 0.37
CYP1A2 P05177 1/20 0.37
GRM1 Q13255 1/20 0.37
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28363838 0.82 CYP1A2 (0.52) KDM4EALDH1A1HPGDCYP3A4KMT2A
SCHEMBL400759 0.80 NOTUM (0.43) CYP3A4CYP2C9KMT2AHAAONOTUM
SCHEMBL3107355 0.79 NOTUM (0.40) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL1478873 0.77 TDP1 (0.44) KDM4EALDH1A1HPGDHSD17B10HAAO
SCHEMBL398481 0.76 RXRB (0.44) KDM4EALDH1A1HPGDHSD17B10HAAO
SCHEMBL9943824 0.76 GRIA4 (0.50) KDM4EALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL857301 0.76 ALDH1A1 (0.65) KDM4EALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL30083685 0.76 ALDH1A1 (0.65) KDM4EALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL1352723 0.76 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL2650251 0.74 CSNK2A1 (0.44) ALDH1A1KMT2ASELLSELPMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968579-A1 PHARMACEUTICAL COMPOUNDS Astex Therapeutics Limited (GB) 2008-09-17 EP disclosed
WO-2007077435-A1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2007-07-12 WO disclosed