SCHEMBL5255462

SCHEMBL5255462

C=CCONC1CN(C(=O)C(F)(F)F)C(C(=O)O)c2cccc(OCc3ccccc3)c21

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KDM1A O60341 2/20 0.35
MRGPRX4 Q96LA9 3/20 0.34
NPC1 O15118 1/20 0.33
S1PR5 Q9H228 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187180 0.91 KMT2A (0.38) HTR1ASLC6A2SLC6A4SLC6A3SIRT1
SCHEMBL4696919 0.83 MEN1 (0.36) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL5253702 0.77 HTR1A (0.38) HTR1ASLC6A2SLC6A4SLC6A3KDM1A
SCHEMBL5252503 0.75 MRGPRX4 (0.33) MRGPRX4S1PR5
SCHEMBL4144345 0.74 MEN1 (0.38)
SCHEMBL5185631 0.72 KMT2A (0.39) HTR1ASLC6A2SLC6A4SLC6A3MRGPRX4
SCHEMBL4696338 0.72 MEN1 (0.33)
SCHEMBL5253676 0.72 ACE (0.36)
SCHEMBL5255876 0.70 MEN1 (0.37) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL5255804 0.70 ALOX15 (0.36) KDM1AMRGPRX4S1PR5SIRT1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed
EP-1399444-A2 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS Aventis Pharma S.A. (FR) 2004-03-24 EP disclosed
WO-2002100860-A2 HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-12-19 WO disclosed