SCHEMBL4696924

SCHEMBL4696924

CC(=O)N1CCN(Cc2ccc(C(=O)N(C)CCOC(=O)N(c3ccccc3-c3ccccc3)N3CC[CH]CC3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
ACHE P22303 2/20 0.39
MCHR1 Q99705 2/20 0.38
BCHE P06276 1/20 0.37
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
KDR P35968 1/20 0.36
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692594 0.92 CHRM2 (0.42) CHRM2ACHEMCHR1BCHEPOLB
SCHEMBL4694973 0.92 MCHR1 (0.40) CHRM2HRH3ACHEMCHR1BCHE
SCHEMBL4693819 0.90 CHRM2 (0.42) CHRM2HRH3ACHEMCHR1BCHE
SCHEMBL5280124 0.89 CHRM2 (0.46) CHRM2ACHEMCHR1BCHEPDCD1
SCHEMBL6021912 0.87 CHRM2 (0.56) CHRM2ACHEBCHECD274
SCHEMBL4692420 0.85 MCHR1 (0.38) CHRM2ACHEMCHR1BCHEPOLB
SCHEMBL4695275 0.82 CHRM2 (0.35) CHRM2HRH3MCHR1
SCHEMBL5273742 0.79 NAMPT (0.35) CHRM2CD274LMNA
SCHEMBL4693546 0.77 POLB (0.40) ACHEBCHELMNAPOLB
SCHEMBL4695712 0.77 MEN1 (0.38) HRH3MCHR1PDCD1CD274KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP claimed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO claimed
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP disclosed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO disclosed