SCHEMBL4697072

SCHEMBL4697072

CC(C)(C)S(=O)(=O)CCCOC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.39
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
CHRM5 P08912 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
HTR1A P08908 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHRNA7 P36544 1/20 0.39
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CA2 P00918 2/20 0.33
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4699116 0.88 LMNA (0.42) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL4698460 0.78 LMNA (0.43) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL9883759 0.75 CACNA1H (0.33) CYP2C19CA2CACNA1H
SCHEMBL28431194 0.75 LMNA (0.41) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL28179923 0.75 APP (0.46) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL27029803 0.74 LMNA (0.40) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL29271182 0.74 LMNA (0.40) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL12247474 0.73 CYP3A4 (0.31) TSHR
SCHEMBL13617276 0.71 ALOX15 (0.48) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL2746597 0.71 TSHR (0.52) LMNACHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987037-A2 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-11-05 EP disclosed
WO-2007097470-A2 FUSED NITROGEN- COMPRISING HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-30 WO disclosed