SCHEMBL4697511

SCHEMBL4697511

Cc1sc(C)c(C(=O)N2CC3CN([C](CC(N)=O)c4ccccc4)C[C@H]3C2)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.41
MAPT P10636 6/20 0.41
LMNA P02545 3/20 0.41
CCR5 P51681 3/20 0.41
HPGD P15428 6/20 0.41
PLA2G1B P04054 1/20 0.41
MAPK1 P28482 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GAA P10253 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229656 0.78 CCR5 (0.40) CCR5
SCHEMBL4690328 0.75 CCR5 (0.52) CCR5
SCHEMBL4695956 0.68 HCRTR1 (0.37) CCR5HPGDHCRTR1HCRTR2
SCHEMBL4690325 0.68 CCR5 (0.40) CCR5
SCHEMBL4691448 0.65 CCR5 (0.50) CCR5
SCHEMBL5237889 0.62 HCRTR1 (0.53) CCR5HCRTR1HCRTR2
SCHEMBL5232470 0.61 CCR5 (0.54) CCR5HCRTR1HCRTR2
SCHEMBL5232788 0.61 CHRNB2 (0.44) MAPTLMNAMAPK1MEN1KMT2A
SCHEMBL4696789 0.61 CCR5 (0.57) CCR5HCRTR1HCRTR2
SCHEMBL14676930 0.60 CHRNB2 (0.71) ALDH1A1HPGDPLA2G1BATG4BHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed