SCHEMBL4698323

SCHEMBL4698323

COCC(COCCOC(N)=O)OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
CHRM5 P08912 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
LMNA P02545 2/20 0.38
HTR1A P08908 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
AKT1 P31749 3/20 0.36
AKT2 P31751 3/20 0.36
AKT3 Q9Y243 3/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28565968 0.84 ALOX15 (0.41) CHRNB2CHRNA4CHRM2CHRM4CHRM5
SCHEMBL4700322 0.79 CHRNB2 (0.43) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL20784046 0.78 ALOX15 (0.46) CHRNB2CHRNA4CHRM2CHRM4CHRM5
SCHEMBL10821810 0.77 LPAR1 (0.43) ALDH1A1AKT1AKT2AKT3PIK3R1
SCHEMBL11806933 0.76 CHRNB2 (0.47) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL29221545 0.76 TSHR (0.46) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL30678661 0.76 TSHR (0.46) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL631206 0.76 TSHR (0.46) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL5531906 0.76 TSHR (0.46) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4
SCHEMBL4698121 0.75 HSD17B10 (0.50) ALDH1A1CHRNB2CHRNA4CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987037-A2 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-11-05 EP disclosed
WO-2007097470-A2 FUSED NITROGEN- COMPRISING HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-30 WO disclosed