SCHEMBL4698619

SCHEMBL4698619

O=c1[nH]c2ccccc2n1C1CCN(C(=S)NC(Cc2ccccc2)c2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 7/20 0.58
OPRM1 P35372 3/20 0.55
OPRK1 P41145 1/20 0.55
OPRL1 P41146 1/20 0.55
CYP3A4 P08684 1/20 0.53
ALDH1A1 P00352 2/20 0.50
MAPK1 P28482 1/20 0.50
RAMP1 O60894 1/20 0.49
CHRM2 P08172 2/20 0.48
CHRM4 P08173 2/20 0.48
CHRM1 P11229 2/20 0.48
CHRM5 P08912 1/20 0.48
CHRM3 P20309 1/20 0.48
HSD11B1 P28845 1/20 0.48
PLD2 O14939 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698559 0.86 CALCRL (0.65) CALCRLOPRM1OPRK1OPRL1CYP3A4
SCHEMBL4698557 0.86 CALCRL (0.65) CALCRLOPRM1OPRK1OPRL1CYP3A4
SCHEMBL12658316 0.77 CHRM1 (0.61) OPRM1OPRK1OPRL1ALDH1A1MAPK1
SCHEMBL13101545 0.77 OPRM1 (0.57) CALCRLOPRM1OPRK1OPRL1ALDH1A1
SCHEMBL1832853 0.76 OPRM1 (0.52) CALCRLOPRM1OPRK1OPRL1CYP3A4
SCHEMBL1832858 0.76 OPRM1 (0.52) CALCRLOPRM1OPRK1OPRL1CYP3A4
SCHEMBL22588021 0.75 OPRK1 (0.67) CALCRLOPRM1OPRK1OPRL1CYP3A4
SCHEMBL1833332 0.74 HSD11B1 (0.68) OPRM1OPRK1OPRL1ALDH1A1MAPK1
SCHEMBL1760919 0.73 HSD11B1 (0.67) OPRM1OPRK1OPRL1ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL3106327 0.73 HSD11B1 (0.67) OPRM1OPRK1OPRL1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1330451-B1 SUBSTITUTED BENZIMIDAZOL-2-ONES AS VASOPRESSIN RECEPTOR ANTAGONISTS AND NEUROPEPTIDE Y MODULATORS ORTHO MCNEIL PHARM INC (US) 2008-01-23 EP claimed