SCHEMBL4698962

SCHEMBL4698962

CC(C)C[C@@H](C(N)=O)N(CC#N)c1nscc1-c1cnc(N2CCNCC2)nc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.37
CTSS P25774 10/20 0.37
CTSB P07858 9/20 0.37
CTSK P43235 8/20 0.37
RET P07949 2/20 0.33
FEN1 P39748 1/20 0.33
ALDH1A1 P00352 2/20 0.31
CYP1A2 P05177 2/20 0.31
HPGD P15428 2/20 0.31
CASP1 P29466 2/20 0.31
CASP7 P55210 2/20 0.31
HSD17B10 Q99714 2/20 0.31
MEN1 O00255 1/20 0.31
CYP2C9 P11712 1/20 0.31
KMT2A Q03164 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
GPR119 Q8TDV5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704327 0.87 CTSL (0.51) CTSLCTSSCTSBCTSK
SCHEMBL4701851 0.85 CTSL (0.49) CTSLCTSSCTSBCTSK
SCHEMBL4698882 0.79 CTSL (0.42) CTSLCTSSCTSBCTSK
SCHEMBL4703890 0.77 CTSS (0.40) CTSLCTSSCTSBCTSKALDH1A1
SCHEMBL4705295 0.76 CTSL (0.45) CTSLCTSSCTSBCTSKRET
SCHEMBL4704891 0.75 CTSL (0.37) CTSLCTSSCTSBCTSK
SCHEMBL4698649 0.74 CTSL (0.48) CTSLCTSSCTSBCTSK
SCHEMBL4703666 0.73 CTSL (0.47) CTSLCTSSCTSBCTSKRET
SCHEMBL5872529 0.73 CTSL (0.47) CTSLCTSSCTSBCTSKRET
SCHEMBL4698985 0.73 CTSL (0.57) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed