SCHEMBL4704891

SCHEMBL4704891

CC(C)C[C@@H](C(N)=O)N(CC#N)c1nscc1-c1ccc(N2CC(C)NC(C)C2)cc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.37
CTSB P07858 5/20 0.37
CTSS P25774 5/20 0.37
CTSK P43235 4/20 0.37
GHSR Q92847 5/20 0.32
TGFBR1 P36897 1/20 0.32
ACVR1 Q04771 1/20 0.32
KCNH2 Q12809 1/20 0.32
MLNR O43193 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704327 0.86 CTSL (0.51) CTSLCTSBCTSSCTSKTGFBR1
SCHEMBL4703890 0.84 CTSS (0.40) CTSLCTSBCTSSCTSKTGFBR1
SCHEMBL4701851 0.84 CTSL (0.49) CTSLCTSBCTSSCTSKTGFBR1
SCHEMBL4703605 0.78 MEN1 (0.31)
SCHEMBL4703744 0.77 KDM4E (0.36) CTSLCTSBCTSSCTSK
SCHEMBL4703503 0.77 KDM4E (0.36) CTSLCTSBCTSSCTSK
SCHEMBL4698962 0.75 CTSL (0.37) CTSLCTSBCTSSCTSK
SCHEMBL4700189 0.74 CTSL (0.57) CTSLCTSBCTSSCTSK
SCHEMBL4698882 0.74 CTSL (0.42) CTSLCTSBCTSSCTSK
SCHEMBL4698649 0.73 CTSL (0.48) CTSLCTSBCTSSCTSKTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed