SCHEMBL469936

SCHEMBL469936

CCOc1ccc(-c2ccc(C(C)C(=O)Nc3cc(C)nn3C)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.47
FFAR1 O14842 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ACACB O00763 5/20 0.45
ACACA Q13085 2/20 0.45
MAPT P10636 1/20 0.43
TSHR P16473 2/20 0.42
RAB9A P51151 1/20 0.42
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CACNA1H O95180 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL462647 0.91 ACACB (0.50) FFAR1MEN1KMT2AACACB
SCHEMBL1822727 0.78 FAAH (0.58) PTGS2MAPTRAB9ASMN1; SMN2AKR1C3
SCHEMBL12677082 0.72 MTNR1B (0.56) MEN1KMT2AMAPTTSHRRAB9A
SCHEMBL1819860 0.68 MAPT (0.62) PTGS2MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL16214695 0.68 SMN1; SMN2 (0.60) ACACBMAPTTSHRRAB9ASMN1; SMN2
SCHEMBL16214700 0.68 ACACB (0.64) ACACB
SCHEMBL27513384 0.67 AKR1C3 (0.57) PTGS2ACACBACACATSHRAKR1C3
SCHEMBL13255719 0.67 SMN1; SMN2 (0.61) MEN1KMT2ATSHRRAB9ASMN1; SMN2
SCHEMBL16214701 0.66 ACACB (0.57) ACACBRAB9A
SCHEMBL5881684 0.66 AKR1C3 (0.73) PTGS2ACACBTSHRAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012032014-A1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-03-15 WO disclosed