SCHEMBL4699759

SCHEMBL4699759

O=C(NCc1ncc(C(=O)O)cc1Cl)NC1c2ccccc2CCC2C=CC=CC21

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 5/20 0.36
TAS1R1 Q7RTX1 5/20 0.36
TAS1R2 Q8TE23 4/20 0.36
ALDH1A1 P00352 1/20 0.35
EPHX2 P34913 4/20 0.34
OPRM1 P35372 2/20 0.34
OPRK1 P41145 2/20 0.34
OPRL1 P41146 1/20 0.34
DHODH Q02127 1/20 0.34
P2RX7 Q99572 1/20 0.33
NTRK1 P04629 2/20 0.32
BACE1 P56817 1/20 0.32
HPGDS O60760 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701668 0.81 ALDH1A1 (0.39) TAS1R3TAS1R1ALDH1A1EPHX2OPRM1
SCHEMBL4702800 0.72 KMT2A (0.40) TAS1R3TAS1R1ALDH1A1OPRM1OPRK1
SCHEMBL4702365 0.70 OPRM1 (0.34) TAS1R3TAS1R1ALDH1A1OPRM1OPRK1
SCHEMBL6387406 0.68 ALDH1A1 (0.47) TAS1R3TAS1R1ALDH1A1HPGDS
SCHEMBL4758046 0.65 EPHX2 (0.49) TAS1R3TAS1R1ALDH1A1EPHX2OPRM1
SCHEMBL4756002 0.63 ALDH1A1 (0.39) TAS1R3TAS1R1TAS1R2ALDH1A1OPRM1
SCHEMBL6388815 0.63 ALDH1A1 (0.36) TAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL6388812 0.63 ALDH1A1 (0.36) TAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL6389721 0.62 ROCK2 (0.37) ALDH1A1
SCHEMBL4704630 0.60 ALDH1A1 (0.38) TAS1R3TAS1R1ALDH1A1P2RX7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458684-B1 THERAPEUTIC HETEROCYCLES AS BRADYKININ B2 RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2008-01-16 EP disclosed