SCHEMBL4699896

SCHEMBL4699896

CCOc1cc(CN(c2ncc(C#N)c(N)n2)C2CCNCC2)cc(OCOC)c1I

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 8/20 0.37
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
SLC6A3 Q01959 3/20 0.34
NOS2 P35228 6/20 0.32
NOS3 P29474 5/20 0.32
NOS1 P29475 5/20 0.32
FGFR4 P22455 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703961 0.86 IKBKB (0.40) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4703405 0.86 IKBKB (0.40) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4700035 0.86 IKBKB (0.40) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4705848 0.85 SLC6A2 (0.41) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4701133 0.84 SLC6A2 (0.42) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4702963 0.83 SLC6A2 (0.41) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4704338 0.83 SLC6A2 (0.41) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4701500 0.83 SLC6A2 (0.41) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4703002 0.82 DHFR (0.43) IKBKBSLC6A2SLC6A4SLC6A3NOS2
SCHEMBL4705830 0.78 IKBKB (0.35) IKBKBSLC6A2SLC6A4SLC6A3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed