SCHEMBL4701133

SCHEMBL4701133

CCOc1cc(CN(c2ncc(C#N)c(N)n2)C2CCNCC2)ccc1C

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.42
SLC6A4 P31645 5/20 0.42
SLC6A3 Q01959 5/20 0.42
IKBKB O14920 7/20 0.41
NOS2 P35228 6/20 0.36
NOS3 P29474 5/20 0.36
NOS1 P29475 5/20 0.36
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
SSTR5 P35346 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705848 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4704338 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4701500 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4703961 0.89 IKBKB (0.40) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4700035 0.89 IKBKB (0.40) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4703405 0.89 IKBKB (0.40) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4702963 0.86 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4703002 0.85 DHFR (0.43) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4699896 0.84 IKBKB (0.37) SLC6A2SLC6A4SLC6A3IKBKBNOS2
SCHEMBL4705855 0.84 IKBKB (0.42) SLC6A2SLC6A4SLC6A3IKBKBNOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed