SCHEMBL4701291

SCHEMBL4701291

NC(=O)C1Cc2ccccc2C1c1nccs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.43
NOS2 P35228 1/20 0.43
GRM1 Q13255 1/20 0.37
GAA P10253 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SLC9A3 P48764 1/20 0.35
RBP4 P02753 1/20 0.34
NR3C1 P04150 5/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PGR P06401 2/20 0.33
AR P10275 2/20 0.33
NPC1 O15118 1/20 0.33
METAP2 P50579 1/20 0.33
RAB9A P51151 1/20 0.33
METAP1 P53582 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ESR1 P03372 1/20 0.33
GPR88 Q9GZN0 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701188 0.83 CHEK2 (0.35) NOS3NOS2ALDH1A1LMNASMN1; SMN2
SCHEMBL28234105 0.72 HTR2A (0.39) GAAALDH1A1LMNA
SCHEMBL28235060 0.70 PRCP (0.40) GAAALDH1A1
SCHEMBL2038839 0.69 GPR88 (0.42) NOS3NOS2GRM1ALDH1A1GPR88
SCHEMBL4283036 0.69 ALDH1A1 (0.41) GAAALDH1A1
SCHEMBL4283038 0.69 KDM1A (0.42) GAAALDH1A1
SCHEMBL4286040 0.69 KDM1A (0.42) GAAALDH1A1
SCHEMBL4286038 0.69 ALDH1A1 (0.41) GAAALDH1A1
SCHEMBL28127659 0.69 ALDH1A1 (0.41) GAAALDH1A1
SCHEMBL28176111 0.67 NOS3 (0.67) NOS3NOS2LMNASMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973890-A2 INDANE MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-KB ACTIVITY AND USE THEREOF Brystol-Myers Squibb Company (US) 2008-10-01 EP claimed
WO-2007073503-A2 INDANE MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-KB ACTIVITY AND USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-28 WO claimed