SCHEMBL4701807

SCHEMBL4701807

Cc1nsc(N(CC#N)[C@@H](CC(C)C)C(N)=O)c1-c1ccc(N2CCN(C(C)C)CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.36
ACVR1 Q04771 2/20 0.36
CTSK P43235 12/20 0.35
CTSS P25774 11/20 0.35
CTSL P07711 11/20 0.35
CTSB P07858 11/20 0.35
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
ACVR1B P36896 1/20 0.34
ACVRL1 P37023 1/20 0.34
TNIK Q9UKE5 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
MEN1 O00255 1/20 0.32
ESR1 P03372 1/20 0.32
KMT2A Q03164 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4699905 0.91 CTSS (0.41) TGFBR1ACVR1CTSKCTSSCTSL
SCHEMBL4703327 0.90 CTSL (0.46) ACVR1CTSKCTSSCTSLCTSB
SCHEMBL4703250 0.90 CTSL (0.46) ACVR1CTSKCTSSCTSLCTSB
SCHEMBL4703010 0.89 CTSS (0.37) CTSKCTSSCTSLCTSBESR1
SCHEMBL4701237 0.89 CTSS (0.36) CTSKCTSSCTSLCTSB
SCHEMBL4701723 0.89 KDM4E (0.35) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4699979 0.89 CTSS (0.44) CTSKCTSSCTSLCTSBTNIK
SCHEMBL4702728 0.89 RORC (0.35) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL4703971 0.89 CTSS (0.37) TGFBR1ACVR1CTSKCTSSCTSL
SCHEMBL4702148 0.88 CTSS (0.40) CTSKCTSSCTSLCTSBTNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed