SCHEMBL4701911

SCHEMBL4701911

Fc1cc(I)ccc1N=C=S.S=C(Cl)Cl

nearest known ligand 0.31

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.30
ALDH1A1 P00352 1/20 0.30
NR3C1 P04150 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADRA2A P08913 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
ADRA2C P18825 1/20 0.30
MAOA P21397 1/20 0.30
DRD1 P21728 1/20 0.30
SLC6A4 P31645 1/20 0.30
HTR2B P41595 1/20 0.30
CCR2 P41597 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL990169 0.93 ABCB11 (0.33) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL22108953 0.81 ALOX5AP (0.32)
SCHEMBL22108951 0.79 NAAA (0.34) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL21386576 0.79 NAAA (0.34) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL624867 0.74 CYP3A4 (0.38) ALDH1A1CYP3A4HPGDTDP1
SCHEMBL28232289 0.74
SCHEMBL28371956 0.74 ESR1 (0.37) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL3972524 0.74 IDO1 (0.34) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL30298623 0.74 HTR2B (0.33) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4
SCHEMBL6596126 0.74 HTR2B (0.33) ABCB11ALDH1A1NR3C1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981892-A1 THIENO-PYRIDINE DERIVATIVES AS MEK INHIBITORS UCB Pharma, S.A. (BE) 2008-10-22 EP disclosed
WO-2007088345-A1 THIENO-PYRIDINE DERIVATIVES AS MEK INHIBITORS UCB PHARMA S.A. (BE) 2007-08-09 WO disclosed