SCHEMBL4702177

SCHEMBL4702177

CCOc1cc(CN(c2ncc(C(=O)O)c(C(F)(F)F)n2)C2CCNCC2)ccc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.41
SLC6A2 P23975 3/20 0.39
SLC6A4 P31645 3/20 0.39
SLC6A3 Q01959 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TACR1 P25103 2/20 0.36
KCNH2 Q12809 1/20 0.36
POLB P06746 1/20 0.35
PDE4B Q07343 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703140 0.92 REN (0.43) RENSLC6A2SLC6A4SLC6A3TACR1
SCHEMBL4705277 0.91 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4703017 0.91 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4706291 0.90 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4704752 0.88 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4704998 0.87 KDM4E (0.37) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4704429 0.87 CNR2 (0.37) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL4705287 0.85 TP53 (0.38) SLC6A2SLC6A4SLC6A3TACR1ALDH1A1
SCHEMBL4705237 0.85 TACR1 (0.39) SLC6A2SLC6A4SLC6A3TACR1KCNH2
SCHEMBL3974580 0.84 REN (0.41) RENSLC6A2SLC6A4L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed