SCHEMBL4705237

SCHEMBL4705237

CCOc1cc(CN(c2ncc(C(=O)O)c(C(F)(F)F)n2)C2CCNCC2)cc(OCC)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 1/20 0.35
JUN P05412 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
CNR2 P34972 1/20 0.35
CETP P11597 4/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704752 0.89 SLC6A2 (0.36) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4704599 0.89 SLC6A2 (0.38) TACR1SLC6A2SLC6A4SLC6A3CNR2
SCHEMBL4704429 0.89 CNR2 (0.37) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4704998 0.89 KDM4E (0.37) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4705277 0.85 SLC6A2 (0.40) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4703017 0.85 SLC6A2 (0.40) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4705287 0.85 TP53 (0.38) TACR1SLC6A2SLC6A4SLC6A3JUN
SCHEMBL4706291 0.85 SLC6A2 (0.39) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4702177 0.85 REN (0.41) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4703140 0.78 REN (0.43) TACR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed