SCHEMBL4703740

SCHEMBL4703740

CC(C)C[C@H](N)C(=O)N(CC#N)c1nscc1-c1ccc(C(C)(C)N)cc1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
AAK1 Q2M2I8 2/20 0.32
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4700000 0.88 CTSB (0.34) CTSLCTSSCTSKAAK1
SCHEMBL4702315 0.87 AAK1 (0.33) CTSLCTSSCTSKAAK1
SCHEMBL4703534 0.85 GSK3B (0.33) CTSLCTSSCTSKAAK1
SCHEMBL6209286 0.84 KDM4E (0.36) AAK1
SCHEMBL6209280 0.84 KDM4E (0.36) AAK1
SCHEMBL6208510 0.78 CTSB (0.39) CTSLCTSSCTSKAAK1DPP4
SCHEMBL4701834 0.78 CTSB (0.39) CTSLCTSSCTSKAAK1DPP4
SCHEMBL4701046 0.77 AKR1C3 (0.34) CTSLCTSSCTSKAAK1DPP4
SCHEMBL4700769 0.75 CTSL (0.38) CTSLCTSSCTSK
SCHEMBL4700510 0.70 CTSL (0.48) CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed