SCHEMBL4701046

SCHEMBL4701046

CC(C)C[C@H](N)C(=O)N(CC#N)c1cscc1-c1ccc(C(C)(C)C)cc1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSL P07711 3/20 0.33
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33
CTSB P07858 1/20 0.33
GRIA4 P48058 4/20 0.31
THRB P10828 2/20 0.31
TP53 P04637 1/20 0.31
GRIA2 P42262 3/20 0.31
AAK1 Q2M2I8 1/20 0.31
LGMN Q99538 1/20 0.31
DPP4 P27487 2/20 0.30
GPR88 Q9GZN0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703749 0.86 CTSK (0.32) CTSLCTSSCTSKCTSBAAK1
SCHEMBL4700607 0.82 GPR88 (0.37) MEN1ALDH1A1KMT2ACTSLCTSS
SCHEMBL4701624 0.77 CTSL (0.42) CTSLCTSSCTSBDPP4
SCHEMBL4703740 0.77 CTSL (0.33) CTSLCTSSCTSKAAK1DPP4
SCHEMBL4700000 0.71 CTSB (0.34) ALDH1A1CTSLCTSSCTSKCTSB
SCHEMBL4703612 0.70 CTSS (0.34) CTSLCTSSCTSKCTSB
SCHEMBL4702315 0.70 AAK1 (0.33) CTSLCTSSCTSKCTSBAAK1
SCHEMBL4704688 0.68 CTSL (0.33) CTSLCTSSCTSKCTSBLGMN
SCHEMBL4703534 0.68 GSK3B (0.33) CTSLCTSSCTSKAAK1
SCHEMBL6209286 0.67 KDM4E (0.36) KDM4EALDH1A1CTSBAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed