SCHEMBL4704375

SCHEMBL4704375

Cn1c(SCCCN2CCc3ccc(C(=O)c4ccccc4)cc3C2)nnc1-c1ccsc1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.49
DRD2 P14416 17/20 0.49
KCNH2 Q12809 14/20 0.49
HRH1 P35367 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705240 0.91 DRD3 (0.58) DRD3DRD2KCNH2HRH1
SCHEMBL4702422 0.90 DRD3 (0.47) DRD3DRD2KCNH2
SCHEMBL4701966 0.90 DRD3 (0.56) DRD3DRD2KCNH2HRH1
SCHEMBL4704001 0.88 DRD3 (0.55) DRD3DRD2KCNH2HRH1
SCHEMBL4702317 0.86 DRD3 (0.56) DRD3DRD2KCNH2
SCHEMBL4701331 0.85 DRD3 (0.56) DRD3DRD2KCNH2HRH1
SCHEMBL4706365 0.84 DRD3 (0.57) DRD3DRD2KCNH2HRH1
SCHEMBL4387104 0.83 DRD3 (0.59) DRD3DRD2KCNH2HRH1
SCHEMBL4701336 0.83 DRD3 (0.47) DRD3DRD2KCNH2HRH1
SCHEMBL6192786 0.83 ALDH1A1 (0.53) DRD3DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594861-B1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO KG (DE) 2008-06-18 EP disclosed
EP-1594861-A1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF Abbott GmbH & Co. KG (DE) 2005-11-16 EP disclosed
WO-2004069830-A1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO. KG (DE) 2004-08-19 WO disclosed