SCHEMBL4701331

SCHEMBL4701331

Cn1c(SCCCN2CCc3ccc(C(=O)c4cccc(F)c4)cc3C2)nnc1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 19/20 0.56
DRD2 P14416 15/20 0.56
KCNH2 Q12809 11/20 0.56
HTR1A P08908 1/20 0.49
HRH1 P35367 1/20 0.48
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PPARG P37231 1/20 0.46
KMT2A Q03164 1/20 0.46
NR2E3 Q9Y5X4 1/20 0.46
NCOR2 Q9Y618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705240 0.93 DRD3 (0.58) DRD3DRD2KCNH2HTR1AHRH1
SCHEMBL4702554 0.92 DRD3 (0.54) DRD3DRD2KCNH2ALDH1A1
SCHEMBL4704001 0.91 DRD3 (0.55) DRD3DRD2KCNH2HTR1AHRH1
SCHEMBL4701966 0.89 DRD3 (0.56) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4705218 0.88 DRD3 (0.54) DRD3DRD2KCNH2HRH1
SCHEMBL4387104 0.87 DRD3 (0.59) DRD3DRD2KCNH2HTR1AHRH1
SCHEMBL4702436 0.87 DRD2 (0.55) DRD3DRD2KCNH2ALDH1A1
SCHEMBL4702317 0.86 DRD3 (0.56) DRD3DRD2KCNH2ALDH1A1CYP3A4
SCHEMBL4701185 0.86 DRD3 (0.57) DRD3DRD2KCNH2HTR1AHRH1
SCHEMBL4704375 0.85 DRD3 (0.49) DRD3DRD2KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594861-B1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO KG (DE) 2008-06-18 EP disclosed