SCHEMBL4701966

SCHEMBL4701966

Cn1c(SCCCN2CCc3ccc(C(=O)c4ccccc4)cc3C2)nnc1-c1ccncc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 0.56
DRD2 P14416 9/20 0.56
KCNH2 Q12809 8/20 0.56
ALDH1A1 P00352 2/20 0.52
MAPT P10636 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
HDAC3 O15379 2/20 0.51
PTK2 Q05397 2/20 0.51
HDAC2 Q92769 2/20 0.51
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HDAC1 Q13547 1/20 0.51
LMNA P02545 1/20 0.49
HPGD P15428 1/20 0.49
CDC25A P30304 1/20 0.49
CDC25B P30305 1/20 0.49
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705240 0.95 DRD3 (0.58) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL4704001 0.92 DRD3 (0.55) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL4702317 0.91 DRD3 (0.56) DRD3DRD2KCNH2ALDH1A1CYP3A4
SCHEMBL4704375 0.90 DRD3 (0.49) DRD3DRD2KCNH2HRH1
SCHEMBL4701331 0.89 DRD3 (0.56) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL4387104 0.87 DRD3 (0.59) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL4706365 0.86 DRD3 (0.57) DRD3DRD2KCNH2HRH1
SCHEMBL4701185 0.85 DRD3 (0.57) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL6192786 0.85 ALDH1A1 (0.53) DRD3DRD2KCNH2ALDH1A1MAPT
SCHEMBL4701336 0.85 DRD3 (0.47) DRD3DRD2KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594861-B1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO KG (DE) 2008-06-18 EP disclosed