SCHEMBL4705064

SCHEMBL4705064

CCOc1cc(CN(c2ncc(C(=O)O)cn2)C2CCNCC2)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 9/20 0.45
SLC6A4 P31645 9/20 0.45
SLC6A3 Q01959 8/20 0.45
SSTR5 P35346 3/20 0.41
KCNH2 Q12809 2/20 0.39
TACR1 P25103 3/20 0.38
KIFC1 Q9BW19 1/20 0.36
LPAR1 Q92633 1/20 0.35
LPAR5 Q9H1C0 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701211 0.90 SLC6A4 (0.44) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL3973033 0.89 SSTR5 (0.42) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL4703414 0.86 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL4703982 0.86 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL4705277 0.84 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL3971901 0.82 SSTR5 (0.43) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL4702309 0.80 REN (0.44) SLC6A2SLC6A4SLC6A3RXRA
SCHEMBL1121565 0.80 SSTR5 (0.45) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL4701120 0.80 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3SSTR5KCNH2
SCHEMBL3973372 0.79 RXRA (0.41) SLC6A2SLC6A4SLC6A3KCNH2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed