SCHEMBL4705655

SCHEMBL4705655

Nc1cnnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2N2CCOCC2)c1C(=O)c1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.39
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
RORB Q92753 6/20 0.38
RORC P51449 4/20 0.38
NTRK1 P04629 1/20 0.37
P2RX7 Q99572 1/20 0.36
RAB9A P51151 1/20 0.35
KCNH2 Q12809 2/20 0.34
STAT6 P42226 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
GALR3 O60755 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
NR2F2 P24468 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705422 0.91 AKT1 (0.38) AKT1PIK3CAMTORRORBRORC
SCHEMBL4707556 0.85 RORB (0.39) AKT1PIK3CAMTORRORBRORC
SCHEMBL4708522 0.84 RORB (0.42) RORBRORCSMN1; SMN2
SCHEMBL4708724 0.83 MEN1 (0.34) AKT1PIK3CAMTORRORBRORC
SCHEMBL4705450 0.83 RORB (0.42) AKT1RORBRORC
SCHEMBL4707869 0.82 NTRK1 (0.39) AKT1PIK3CAMTORRORBRORC
SCHEMBL4705167 0.82 NTRK1 (0.34) AKT1PIK3CAMTORRORBRORC
SCHEMBL4705884 0.82 RORB (0.40) RORBRORCSMN1; SMN2
SCHEMBL4708031 0.81 NTRK1 (0.34) AKT1PIK3CAMTORRORBRORC
SCHEMBL4705910 0.81 RORB (0.39) RORBRORCGALR3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed