SCHEMBL4708031

SCHEMBL4708031

O=C(c1ccccc1Cl)c1c(CCO)noc1-c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1N1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.34
TACR1 P25103 2/20 0.34
AKT1 P31749 1/20 0.33
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
P2RX7 Q99572 1/20 0.33
RORC P51449 4/20 0.33
RORB Q92753 4/20 0.33
RAB9A P51151 2/20 0.32
PIK3C2B O00750 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32
ALDH1A1 P00352 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705167 0.95 NTRK1 (0.34) NTRK1TACR1AKT1PIK3CAMTOR
SCHEMBL4705298 0.88 RORB (0.36) TACR1P2RX7RORCRORBTHRB
SCHEMBL4706174 0.85 ALDH1A1 (0.33) NTRK1TACR1KMT2AIDO1TDO2
SCHEMBL4708167 0.85 RORB (0.36) TACR1RORCRORBTSHRALDH1A1
SCHEMBL4706589 0.84 TACR1 (0.37) TACR1RORCRORBALDH1A1
SCHEMBL4708724 0.83 MEN1 (0.34) NTRK1TACR1AKT1PIK3CAMTOR
SCHEMBL4708201 0.82 TSHR (0.35) NTRK1MEN1POLBTSHRKMT2A
SCHEMBL4707556 0.82 RORB (0.39) NTRK1AKT1PIK3CAMTORP2RX7
SCHEMBL4705655 0.81 AKT1 (0.39) NTRK1AKT1PIK3CAMTORP2RX7
SCHEMBL4705422 0.81 AKT1 (0.38) NTRK1AKT1PIK3CAMTORP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed