SCHEMBL4705658

SCHEMBL4705658

O=C(CCCN1CCCC(COc2ccccc2C(=O)O)C1)c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.53
HTR2A P28223 1/20 0.52
DRD3 P35462 3/20 0.51
DRD4 P21917 1/20 0.51
CHRNB4 P30926 2/20 0.50
CHRNA3 P32297 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
CHRM2 P08172 1/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
DRD1 P21728 1/20 0.48
ADRA1A P35348 1/20 0.48
OPRM1 P35372 1/20 0.48
KCNH2 Q12809 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054675 0.92 CHRNB4 (0.53) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4051310 0.92 ALDH1A1 (0.51) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4051698 0.91 ALDH1A1 (0.50) DRD2HTR2ADRD3CHRNB4CHRNA3
SCHEMBL4045253 0.90 ALDH1A1 (0.49) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4046290 0.89 ALDH1A1 (0.48) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4048079 0.88 ADRA1A (0.48) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4048748 0.86 DRD2 (0.49) DRD2HTR2ADRD3DRD4CHRNB4
SCHEMBL4046282 0.85 ALDH1A1 (0.50) DRD2HTR2ADRD3DRD4MEN1
SCHEMBL4052789 0.85 DRD2 (0.50) DRD2HTR2ADRD3DRD4MEN1
SCHEMBL4049282 0.84 DRD2 (0.48) DRD2HTR2ADRD3DRD4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421070-B1 NEW PIPERIDINYL DERIVATES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY ASTRAZENECA AB (SE) 2008-11-26 EP claimed