SCHEMBL4706152

SCHEMBL4706152

O=C(NCc1ccccc1Cl)c1nnn(Cc2cc(Cl)cc(Cl)c2)c1N1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.47
MAPT P10636 6/20 0.47
POLB P06746 3/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
THRB P10828 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
HSP90AA1 P07900 1/20 0.44
RAB9A P51151 1/20 0.44
KCNH2 Q12809 1/20 0.44
TSHR P16473 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
GAA P10253 1/20 0.44
CYP2C19 P33261 1/20 0.44
SCN2A Q99250 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708394 0.89 RXFP1 (0.44) RXFP1MAPTPOLBLMNATP53
SCHEMBL4705251 0.82 MAPT (0.52) MAPTPOLBLMNATP53KMT2A
SCHEMBL5796761 0.79 KCNH2 (0.44) POLBSMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL4705947 0.79 MAPT (0.44) MAPTPOLBTP53SMN1; SMN2KCNH2
SCHEMBL4707435 0.78 TP53 (0.44) MAPTPOLBLMNATP53KMT2A
SCHEMBL4707117 0.78 TACR1 (0.45) MAPTPOLBLMNATP53KMT2A
SCHEMBL4707175 0.77 MAPT (0.46) MAPTPOLBLMNATP53KMT2A
SCHEMBL4705003 0.74 ALDH1A1 (0.40) POLBTP53KMT2AMEN1SMN1; SMN2
SCHEMBL4706712 0.71 TP53 (0.52) MAPTPOLBLMNATP53KMT2A
SCHEMBL6480543 0.70 ALDH1A1 (0.36) MAPTTP53SMN1; SMN2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed