SCHEMBL4706771

SCHEMBL4706771

OC(c1ccccc1Cl)c1nccnc1I

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGFBP3 P17936 1/20 0.41
CYP2C19 P33261 2/20 0.40
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
AOC3 Q16853 1/20 0.35
CYP19A1 P11511 1/20 0.35
ACHE P22303 1/20 0.35
CYP2D6 P10635 2/20 0.34
NFKB1 P19838 1/20 0.34
HIF1A Q16665 1/20 0.34
BLM P54132 1/20 0.33
F2RL1 P55085 2/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
KCNA5 P22460 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29976363 0.73 ADRB2 (0.48) IGFBP3CYP2C19ADRB2ADRB1AOC3
SCHEMBL230382 0.73 ADRB2 (0.48) IGFBP3CYP2C19ADRB2ADRB1AOC3
SCHEMBL8745972 0.70 HPGD (0.53) IGFBP3CYP2C19HPGDHSD17B10KDM4C
SCHEMBL4015279 0.69 IGFBP3 (0.43) IGFBP3CYP2C19HPGDHSD17B10KDM4C
SCHEMBL4707217 0.68 CYP2C19 (0.45) IGFBP3CYP2C19HPGDHSD17B10KDM4C
SCHEMBL2901635 0.68 CYP2C19 (0.45) IGFBP3CYP2C19HPGDHSD17B10KDM4C
SCHEMBL4707443 0.67 IGFBP3 (0.39) IGFBP3CYP2C19HPGDHSD17B10KDM4C
SCHEMBL21885163 0.67 KMT2A (0.47) IGFBP3CYP2C19HSD17B10ACHECYP1A2
SCHEMBL11606505 0.66 TSHR (0.50) CYP2C19ADRB2ADRB1AOC3CYP2D6
SCHEMBL477602 0.66 ACP3 (0.53) IGFBP3CYP2C19ADRB2ADRB1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1312136-C Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1646502-A Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2005-07-27 CN disclosed