SCHEMBL4706897

SCHEMBL4706897

CNC1CN(C(I)(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 2/20 0.38
CYP2B6 P20813 1/20 0.35
HRH4 Q9H3N8 3/20 0.34
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
CHRM3 P20309 1/20 0.30
LMNA P02545 1/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
SLC6A3 Q01959 2/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4594764 0.80 GRIN2B (0.38) CYP2B6KDM1AMAOBATML3MBTL1
SCHEMBL11111197 0.77 ALDH1A1 (0.41) KCNN4
SCHEMBL3346414 0.77 LMNA (0.35) CYP2B6ATML3MBTL1CHRM3LMNA
Hydrochloric Acid SCHEMBL11044496 0.76 LMNA (0.38) CYP2B6ATML3MBTL1CHRM3LMNA
SCHEMBL11006008 0.71 CHRM3 (0.48) CHRM3SLC6A2SLC6A4SLC6A3
SCHEMBL19613954 0.70 CYP2B6 (0.51) KCNN4CYP2B6HRH4ATML3MBTL1
SCHEMBL19613953 0.70 CYP2B6 (0.51) KCNN4CYP2B6HRH4ATML3MBTL1
Hydrochloric Acid SCHEMBL6529786 0.69 BPTF (0.35) LMNACYP2D6
SCHEMBL21965412 0.68 BPTF (0.48) HRH4KDM1AMAOBSIGMAR1L3MBTL1
SCHEMBL31214046 0.68 CYP2B6 (0.59) CYP2B6SIGMAR1CHRM3LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991550-A1 AMINO PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS Cellzome Limited (GB) 2008-11-19 EP disclosed
EP-1860109-A1 Azetidine amino pyrimidine compounds for the treatment of inflammatory disorders Cellzome (UK) Ltd. (GB) 2007-11-28 EP disclosed
WO-2007090854-A1 AZETIDINE AMINO PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS CELLZOME (UK) LTD. (GB) 2007-08-16 WO disclosed
WO-2007090852-A1 AMINO PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS CELLZOME LIMITED (GB) 2007-08-16 WO disclosed