SCHEMBL4594764

SCHEMBL4594764

IC(c1ccccc1)(c1ccccc1)N1CC(NC2CC2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.38
KDM1A O60341 11/20 0.33
MAOB P27338 6/20 0.33
MAOA P21397 3/20 0.33
LMNA P02545 2/20 0.33
SLC6A4 P31645 2/20 0.33
CISD1 Q9NZ45 1/20 0.33
KDM1B Q8NB78 1/20 0.33
RCOR1 Q9UKL0 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
SCN1A P35498 1/20 0.33
KMT2A Q03164 1/20 0.33
SCN2A Q99250 1/20 0.33
SCN3A Q9NY46 1/20 0.33
CCR2 P41597 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706897 0.80 KCNN4 (0.38) KDM1AMAOBLMNASLC6A4SLC6A2
SCHEMBL3346414 0.76 LMNA (0.35) LMNAMEN1CYP2D6HRH1SCN1A
Hydrochloric Acid SCHEMBL11044496 0.74 LMNA (0.38) LMNAMEN1CYP2D6HRH1SCN1A
SCHEMBL11006008 0.70 CHRM3 (0.48) GRIN2BSLC6A4SLC6A2HRH1
SCHEMBL11111197 0.69 ALDH1A1 (0.41)
Hydrochloric Acid SCHEMBL6529786 0.68 BPTF (0.35) LMNAMEN1CYP2D6HRH1SCN1A
SCHEMBL31214046 0.67 CYP2B6 (0.59) GRIN2BLMNAHTR2AMEN1CYP2D6
SCHEMBL6025470 0.66 CYP2B6 (0.34) MEN1KMT2ACYP2B6
SCHEMBL4594663 0.66 L3MBTL3 (0.45) GRIN2BHTR2AMEN1CYP2D6HRH1
Hydrochloric Acid SCHEMBL8942152 0.64 L3MBTL3 (0.44) GRIN2BHTR2AMEN1CYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945646-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS Cellzome (UK) Ltd. (GB) 2008-07-23 EP disclosed
WO-2007039467-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS CELLZOME (UK) LTD. (GB) 2007-04-12 WO disclosed