SCHEMBL4706969

SCHEMBL4706969

O=C(NCc1ccccc1Br)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 7/20 0.49
CACNA1H O95180 7/20 0.49
TACR1 P25103 7/20 0.45
CACNA1I Q9P0X4 2/20 0.45
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
TP53 P04637 1/20 0.43
IDH1 O75874 1/20 0.42
CYP19A1 P11511 1/20 0.42
PTGER4 P35408 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707843 0.90 EPHX2 (0.48) CACNA1GCACNA1HTACR1ALDH1A1GAA
SCHEMBL4705917 0.89 IDH1 (0.50) CACNA1GCACNA1HTACR1ALDH1A1GAA
SCHEMBL4706714 0.89 TACR1 (0.48) CACNA1GCACNA1HTACR1ALDH1A1GAA
SCHEMBL4707735 0.88 TACR1 (0.52) TACR1ALDH1A1GAATP53IDH1
SCHEMBL4707944 0.86 IDH1 (0.48) CACNA1GCACNA1HTACR1ALDH1A1GAA
SCHEMBL4706967 0.85 POLB (0.50) TACR1ALDH1A1GAAIDH1PTGER4
SCHEMBL4708123 0.84 TP53 (0.49) CACNA1GCACNA1HTACR1TP53IDH1
SCHEMBL4706587 0.83 IDH1 (0.52) CACNA1GCACNA1HALDH1A1GAATP53
SCHEMBL4708362 0.81 ALDH1A1 (0.56) ALDH1A1GAATP53CYP19A1
SCHEMBL4706658 0.81 IDH1 (0.62) CACNA1GCACNA1HTACR1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed