SCHEMBL4706967

SCHEMBL4706967

O=C(NCc1ccc(F)cc1)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
IDH1 O75874 1/20 0.49
TACR1 P25103 7/20 0.48
PTGER4 P35408 6/20 0.48
HTT P42858 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707735 0.94 TACR1 (0.52) IDH1TACR1PTGER4HTTALDH1A1
SCHEMBL4708123 0.87 TP53 (0.49) IDH1TACR1
SCHEMBL4707843 0.86 EPHX2 (0.48) IDH1TACR1HTTALDH1A1GAA
SCHEMBL4705917 0.85 IDH1 (0.50) POLBIDH1TACR1ALDH1A1GAA
SCHEMBL4706969 0.85 CACNA1G (0.49) IDH1TACR1PTGER4ALDH1A1GAA
SCHEMBL4706714 0.85 TACR1 (0.48) IDH1TACR1ALDH1A1GAA
SCHEMBL4708362 0.83 ALDH1A1 (0.56) ALDH1A1GAA
SCHEMBL4707944 0.83 IDH1 (0.48) IDH1TACR1PTGER4ALDH1A1GAA
SCHEMBL6072058 0.82 ALDH1A1 (0.53) POLBTACR1PTGER4ALDH1A1GAA
SCHEMBL4638473 0.82 ALDH1A1 (0.65) POLBPTGER4ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed