SCHEMBL4707301

SCHEMBL4707301

CCOC(=O)Oc1cc2c(F)cccc2n1CC#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 6/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MAPT P10636 5/20 0.39
TP53 P04637 2/20 0.39
THRB P10828 1/20 0.39
NPSR1 Q6W5P4 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.36
DHODH Q02127 1/20 0.36
MAPK1 P28482 1/20 0.36
STAT3 P40763 1/20 0.36
CCR2 P41597 1/20 0.35
LMNA P02545 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708671 0.89 TDP1 (0.44) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL4706602 0.83 MAPT (0.39) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5623701 0.82 F10 (0.45) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL4707774 0.79 ALDH1A1 (0.38) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL4706772 0.76 MEN1 (0.39) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL4705661 0.75 KDM4E (0.44) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL4706633 0.72 ALOX5 (0.38) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5622537 0.70 ALDH1A1 (0.41) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5623862 0.70 F10 (0.57) TDP1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL5917485 0.68 MAPT (0.46) TDP1ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1625129-B1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT BAYER HEALTHCARE AG (DE) 2008-03-05 EP disclosed
EP-1625129-A1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT Bayer HealthCare AG (DE) 2006-02-15 EP disclosed
WO-2004099212-A1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT BAYER HEALTHCARE AG (DE) 2004-11-18 WO disclosed