SCHEMBL4707650

SCHEMBL4707650

O=C(c1ccccc1Cl)c1ccnnc1-c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORB Q92753 9/20 0.41
RORC P51449 5/20 0.41
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.37
CDC7 O00311 1/20 0.37
ADORA3 P0DMS8 3/20 0.37
PTGER4 P35408 2/20 0.36
GRM2 Q14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708209 0.95 RORB (0.39) RORBRORCCDC7ADORA3GRM2
SCHEMBL4705371 0.93 IDH1 (0.43) RORBRORCGAAGRM2
SCHEMBL4707133 0.92 RORB (0.40) RORBRORCGRM2
SCHEMBL4707172 0.90 RORB (0.46) RORBRORCALDH1A1GAATSHR
SCHEMBL4705502 0.88 RORB (0.39) RORBRORCGAAPTGER4GRM2
SCHEMBL4757295 0.87 RORB (0.51) RORBRORCALDH1A1GAATSHR
SCHEMBL4708690 0.87 RORB (0.40) RORBRORCALDH1A1GAATSHR
SCHEMBL4706528 0.87 RORB (0.36) RORBRORCGRM2
SCHEMBL4705450 0.85 RORB (0.42) RORBRORCALDH1A1GAATSHR
Tradipitant SCHEMBL2898629 0.85 RORB (0.42) RORBRORCCDC7GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed