SCHEMBL4708690

SCHEMBL4708690

Cc1cc(C(=O)c2ccccc2Cl)c(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2ccccc2)nn1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORB Q92753 8/20 0.40
RORC P51449 5/20 0.40
CYP19A1 P11511 2/20 0.39
PTGER4 P35408 2/20 0.38
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
TACR1 P25103 3/20 0.37
TSHR P16473 1/20 0.37
CDC7 O00311 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706783 0.94 RORB (0.38) RORBRORCPTGER4GAATACR1
SCHEMBL4707706 0.92 IDH1 (0.42) RORBRORCPTGER4TACR1
SCHEMBL4707207 0.92 RORB (0.40) RORBRORCPTGER4GAATACR1
SCHEMBL4707181 0.89 RORB (0.40) RORBRORCPTGER4ALDH1A1GAA
SCHEMBL4707650 0.87 RORB (0.41) RORBRORCPTGER4ALDH1A1GAA
SCHEMBL4757295 0.87 RORB (0.51) RORBRORCPTGER4ALDH1A1GAA
SCHEMBL4707926 0.86 P2RX7 (0.36) RORBRORCGAATACR1
SCHEMBL4705944 0.86 TACR1 (0.39) RORBRORCPTGER4GAATACR1
SCHEMBL4707172 0.86 RORB (0.46) RORBRORCPTGER4ALDH1A1GAA
SCHEMBL4708285 0.85 CDC7 (0.38) RORBRORCGAATACR1CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed