SCHEMBL4705502

SCHEMBL4705502

Cc1c(-c2nnccc2C(=O)c2ccccc2Cl)nnn1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORB Q92753 10/20 0.39
RORC P51449 5/20 0.39
TACR1 P25103 2/20 0.39
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 1/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 1/20 0.34
PTGER4 P35408 1/20 0.34
P2RX1 P51575 1/20 0.34
P2RX4 Q99571 1/20 0.34
P2RX7 Q99572 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
GRM2 Q14416 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759328 0.90 RORB (0.43) RORBRORCTACR1KDM4EHTT
SCHEMBL4707181 0.88 RORB (0.40) RORBRORCTACR1KDM4EHTT
SCHEMBL4707650 0.88 RORB (0.41) RORBRORCGAAPTGER4GRM2
SCHEMBL4708209 0.86 RORB (0.39) RORBRORCTACR1GRM2
SCHEMBL4705184 0.86 TACR1 (0.44) RORBRORCTACR1
SCHEMBL4708293 0.85 RORB (0.40) RORBRORCTACR1GAAP2RX7
SCHEMBL4708522 0.85 RORB (0.42) RORBRORCTACR1KDM4EHTT
SCHEMBL4707133 0.85 RORB (0.40) RORBRORCTACR1HTTGRM2
SCHEMBL4705371 0.84 IDH1 (0.43) RORBRORCGAAGRM2
SCHEMBL4706528 0.83 RORB (0.36) RORBRORCTACR1P2RX7GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed