SCHEMBL4708153

SCHEMBL4708153

CN(C)c1c(C(=O)c2c(C=O)noc2-c2ccccc2Cl)nnn1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.39
GPBAR1 Q8TDU6 6/20 0.35
EPAS1 Q99814 2/20 0.33
TACR3 P29371 3/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707521 0.90 TACR1 (0.37) TACR1GPBAR1EPAS1TP53MAPT
SCHEMBL4707071 0.88 TACR1 (0.40) TACR1GPBAR1EPAS1TACR3TP53
SCHEMBL4708775 0.87 TACR1 (0.39) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4637790 0.87 ALDH1A1 (0.43) TACR1
SCHEMBL4709658 0.85 ALDH1A1 (0.38) TACR1GPBAR1
SCHEMBL4705752 0.84 ALDH1A1 (0.33) TACR1EPAS1TACR3MAPTSMN1; SMN2
SCHEMBL4707053 0.82 GPBAR1 (0.34) TACR1GPBAR1
SCHEMBL4638510 0.80 USP2 (0.40) TACR1GPBAR1EPAS1TP53MAPT
SCHEMBL4705246 0.79 TACR1 (0.36) TACR1GPBAR1EPAS1TP53MAPT
SCHEMBL4639421 0.79 ALDH1A1 (0.41) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed