SCHEMBL4708775

SCHEMBL4708775

CN(C)c1c(C(=O)c2c(CCO)noc2-c2ccccc2Cl)nnn1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.39
GPBAR1 Q8TDU6 4/20 0.35
TACR3 P29371 6/20 0.35
TP53 P04637 2/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707071 0.94 TACR1 (0.40) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4705619 0.90 TACR1 (0.36) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4708206 0.90 TACR1 (0.35) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4637802 0.89 TACR1 (0.39) TACR1GPBAR1TACR3TP53GRM2
SCHEMBL4709706 0.87 ALDH1A1 (0.42) TACR1GPBAR1GRM2
SCHEMBL4708153 0.87 TACR1 (0.39) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4706589 0.85 TACR1 (0.37) TACR1GPBAR1GRM2
SCHEMBL4706174 0.84 ALDH1A1 (0.33) TACR1TACR3MAPTSMN1; SMN2GRM2
SCHEMBL4708336 0.84 TACR1 (0.32) TACR1GPBAR1TACR3TP53MAPT
SCHEMBL4758302 0.83 TACR1 (0.37) TACR1GPBAR1TP53MAPTGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed