SCHEMBL4708752

SCHEMBL4708752

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cc(C(F)(F)F)ccc2F)c1-c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORB Q92753 7/20 0.43
IDH1 O75874 1/20 0.42
RORC P51449 4/20 0.39
P2RX7 Q99572 1/20 0.36
CRHR1 P34998 2/20 0.35
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NTRK1 P04629 1/20 0.34
KCNK3 O14649 1/20 0.34
RPS6KA3 P51812 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
KCNA5 P22460 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708468 0.94 RORB (0.41) RORBIDH1RORCP2RX7NTRK1
SCHEMBL4708216 0.92 IDH1 (0.42) RORBIDH1RORCP2RX7CRHR1
SCHEMBL4706699 0.92 RORB (0.42) RORBIDH1RORCP2RX7
SCHEMBL27538912 0.87 RORB (0.44) RORBIDH1RORCSCN5ASCN9A
SCHEMBL4706229 0.87 IDH1 (0.44) RORBIDH1RORCCRHR1SCN5A
SCHEMBL4705528 0.86 RORB (0.43) RORBIDH1RORCP2RX7SCN5A
SCHEMBL4708283 0.86 RORB (0.39) RORBIDH1RORCP2RX7SCN5A
SCHEMBL4706981 0.86 IDH1 (0.42) RORBIDH1RORCCRHR1SCN5A
SCHEMBL4709738 0.85 RORB (0.42) RORBRORCP2RX7CRHR1RPS6KA3
SCHEMBL4708689 0.84 RORB (0.40) RORBIDH1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1312136-C Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2007-04-25 CN disclosed