SCHEMBL4709745

SCHEMBL4709745

Cc1ccc(CNCCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.52
CD274 Q9NZQ7 1/20 0.52
TDP1 Q9NUW8 2/20 0.50
MAPT P10636 1/20 0.50
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CHRM2 P08172 1/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
NPC1 O15118 3/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21066539 0.88 PDCD1 (0.49) PDCD1CD274TDP1CA1CA2
SCHEMBL22452272 0.87 FPR3 (0.47) PDCD1CD274TDP1CA1CA2
SCHEMBL6076877 0.87 HPGD (0.49) PDCD1CD274CA1CA2CHRM2
SCHEMBL12310009 0.87 CA1 (0.47) PDCD1CD274TDP1CA1CA2
SCHEMBL1724201 0.87 GAA (0.60) PDCD1CD274TDP1CA1CA2
SCHEMBL22605044 0.87 ATM (0.58) PDCD1CD274TDP1CA1CA2
SCHEMBL894822 0.87 ATM (0.58) PDCD1CD274TDP1CA1CA2
SCHEMBL5796279 0.86 L3MBTL1 (0.56) TDP1MAPTCA1CA2HDAC1
SCHEMBL21066545 0.86 KMT2A (0.52) CA1CA2CHRM2NPC1L3MBTL1
SCHEMBL22604937 0.86 CD274 (0.53) PDCD1CD274TDP1MAPTCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed