SCHEMBL4710338

SCHEMBL4710338

Cc1ccc(OCCCN(C)C)c(C#Cc2cc(Cl)cc(Cl)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
S1PR4 O95977 6/20 0.40
HRH3 Q9Y5N1 1/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
THPO P40225 1/20 0.37
RAB9A P51151 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HTR1B P28222 1/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710981 0.90 GRM5 (0.47) CYP1A2CYP2D6CYP2C19S1PR4HPGD
SCHEMBL4711351 0.85 S1PR4 (0.41) S1PR4MAPTHPGDNPC1LMNA
SCHEMBL4711565 0.84 HTR1B (0.45) CYP1A2CYP2D6CYP2C19HRH3HPGD
SCHEMBL7348551 0.83 KDM4E (0.42) CYP1A2CYP2D6CYP2C19MAPK1ALDH1A1
SCHEMBL4710329 0.82 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19HTR1B
SCHEMBL4712830 0.82 ALDH1A1 (0.39) CYP1A2CYP2D6CYP2C19MAPK1ALDH1A1
SCHEMBL4710572 0.81 THRA (0.37) CYP1A2CYP2D6CYP2C19HPGDMAPK1
SCHEMBL4712681 0.81 GRM5 (0.42) CYP1A2CYP2D6CYP2C19HTR1B
SCHEMBL4712038 0.78 GRM5 (0.49)
SCHEMBL4713011 0.75 GRM5 (0.49) S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-B1 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2008-04-23 EP claimed
EP-0998459-B1 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2008-04-23 EP disclosed