SCHEMBL7348551

SCHEMBL7348551

CN(C)CCCOc1ccc(C(=O)O)nc1C#Cc1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.42
ALDH1A1 P00352 4/20 0.42
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GAA P10253 2/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
THRA P10827 2/20 0.38
THRB P10828 2/20 0.38
MRGPRX4 Q96LA9 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
PAICS P22234 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349972 0.88 ALDH1A1 (0.46) KDM4EALDH1A1LMNATDP1GAA
SCHEMBL4712830 0.88 ALDH1A1 (0.39) KDM4EALDH1A1LMNATDP1GAA
SCHEMBL4710338 0.83 CYP1A2 (0.41) KDM4EALDH1A1LMNATDP1MAPK1
SCHEMBL4710572 0.81 THRA (0.37) KDM4EALDH1A1LMNATDP1GAA
SCHEMBL4714453 0.77 ALDH1A1 (0.41) KDM4EALDH1A1LMNATDP1GAA
SCHEMBL4715746 0.76 ALDH1A1 (0.44) KDM4EALDH1A1MAPK1KMT2ACYP1A2
SCHEMBL4710981 0.74 GRM5 (0.47) KDM4EALDH1A1MAPK1CYP1A2CYP2D6
SCHEMBL4712903 0.73 HPGD (0.41) ALDH1A1LMNAGAATHRATHRB
SCHEMBL4715224 0.70 ALDH1A1 (0.40) KDM4EALDH1A1LMNATDP1GAA
SCHEMBL4711565 0.70 HTR1B (0.45) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-A2 PYRIDINE DERIVATIVES Novartis AG (CH) 2000-05-10 EP claimed
WO-1999002497-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 1999-01-21 WO claimed