SCHEMBL4715404

SCHEMBL4715404

CCN(C)S(=O)(=O)c1ccc(Cl)c(COCC(=O)c2cccc(C)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.41
HCRTR1 O43613 3/20 0.40
HCRTR2 O43614 3/20 0.40
ALDH1A1 P00352 7/20 0.36
MAPT P10636 5/20 0.36
GAA P10253 2/20 0.35
TSHR P16473 1/20 0.35
GLA P06280 1/20 0.35
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715252 0.85 ALDH1A1 (0.43) VCAM1ALDH1A1MAPTGAALMNA
SCHEMBL4714594 0.85 VCAM1 (0.41) VCAM1HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4713681 0.83 VCAM1 (0.41) VCAM1HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4713390 0.82 VCAM1 (0.46) VCAM1ALDH1A1MAPTGAATSHR
SCHEMBL4714715 0.80 VCAM1 (0.40) VCAM1ALDH1A1MAPTGAATSHR
SCHEMBL4716780 0.80 ALDH1A1 (0.46) ALDH1A1MAPTTSHRLMNAKDM4E
SCHEMBL4713492 0.79 ALDH1A1 (0.46) VCAM1ALDH1A1MAPTTSHRLMNA
SCHEMBL4712737 0.78 ALDH1A1 (0.42) ALDH1A1GAALMNAMAPK1RAB9A
SCHEMBL4713553 0.77 RAB9A (0.53) ALDH1A1MAPTGAATSHRLMNA
SCHEMBL4716110 0.76 NPC1 (0.50) ALDH1A1LMNAMEN1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615904-B1 SUBSTITUTED BENZOSULPHONAMIDES AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA AB (SE) 2008-02-27 EP claimed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US claimed
EP-1615904-A2 SUBSTITUTED BENZOSULPHONAMIDE AS POTENTIATORS OF GLUTAMATE RECEPTORS AstraZeneca AB (SE) 2006-01-18 EP claimed
WO-2004092135-A2 SUBSTITUTED BENZOSULPHONAMIDE AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA (SE) 2004-10-28 WO claimed
EP-1615904-B1 SUBSTITUTED BENZOSULPHONAMIDES AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA AB (SE) 2008-02-27 EP disclosed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US disclosed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US disclosed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US disclosed
EP-1615904-A2 SUBSTITUTED BENZOSULPHONAMIDE AS POTENTIATORS OF GLUTAMATE RECEPTORS AstraZeneca AB (SE) 2006-01-18 EP disclosed
WO-2004092135-A2 SUBSTITUTED BENZOSULPHONAMIDE AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA (SE) 2004-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070021606-A1 Therapeutic compounds GRIN1, GRIN3A, GRM2 VCAM1 1527/4885HCRTR1 284/4885HCRTR2 154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.