SCHEMBL4715993

SCHEMBL4715993

O=C(Cl)CCc1ccc(F)c(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
RIPK1 Q13546 1/20 0.40
FFAR4 Q5NUL3 4/20 0.38
FFAR1 O14842 2/20 0.38
CA2 P00918 1/20 0.37
P2RX7 Q99572 6/20 0.37
CHRNA7 P36544 1/20 0.35
DPP4 P27487 1/20 0.33
FAP Q12884 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31674277 0.85 FFAR4 (0.36) CES2CES1RIPK1FFAR4FFAR1
SCHEMBL23782854 0.84 FFAR4 (0.35) FFAR4FFAR1CHRNA7
SCHEMBL4322411 0.83 CES2 (0.42) CES2CES1RIPK1FFAR4
SCHEMBL4717045 0.82 FFAR1 (0.49) CES2CES1RIPK1FFAR4FFAR1
SCHEMBL30572329 0.81 MPO (0.46) CES2CES1RIPK1FFAR4FFAR1
SCHEMBL5419671 0.80 CES2 (0.43) CES2CES1RIPK1CA2P2RX7
SCHEMBL4718220 0.78 CES2 (0.38) CES2CES1FFAR4FFAR1
SCHEMBL29009960 0.77 HDAC3 (0.47) CES2CES1RIPK1FFAR4FFAR1
Methyl Alcohol SCHEMBL3621979 0.77 RIPK1 (0.43) CES2CES1RIPK1CA2P2RX7
SCHEMBL1477462 0.76 PSEN1 (0.42) CES2CES1RIPK1FFAR4FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337517-B1 PYRIMIDINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 2008-11-26 EP disclosed
EP-1337517-A1 PYRIMIDINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP disclosed
WO-2002030911-A1 PYRIMIDINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM P.L.C. (GB) 2002-04-18 WO disclosed