SCHEMBL4717818

SCHEMBL4717818

CCOC(=O)Oc1c(C)c2c(=O)[nH]cnc2n1-c1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
GAA P10253 3/20 0.38
LMNA P02545 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 4/20 0.38
PDE4B Q07343 3/20 0.38
MAPT P10636 3/20 0.38
TSHR P16473 2/20 0.38
PDE4A P27815 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
HPGD P15428 3/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 2/20 0.36
PPARG P37231 1/20 0.36
NCOA2 Q15596 1/20 0.36
NCOA1 Q15788 1/20 0.36
POLB P06746 1/20 0.35
NLRP3 Q96P20 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721077 0.91 PARP1 (0.37) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL4718967 0.89 KDM4E (0.39) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL4719631 0.89 ALDH1A1 (0.36) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL27614310 0.88 PARP1 (0.38) LMNAMAPTHPGDKMT2APARP1
SCHEMBL291018 0.84 ALDH1A1 (0.44) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL29831878 0.84 ALDH1A1 (0.44) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL4718179 0.84 NPC1 (0.41) ALDH1A1GAALMNAKDM4EHSD17B10
SCHEMBL4718237 0.83 PDE4A (0.40) ALDH1A1GAALMNAKDM4EPDE4B
SCHEMBL4542766 0.78 NOTUM (0.41) LMNAPDE4BMAPTPDE4APDE4C
SCHEMBL29831842 0.77 HPGD (0.42) ALDH1A1GAALMNAKDM4EPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458722-B1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2008-10-15 EP claimed
EP-1458722-B1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2008-10-15 EP disclosed