SCHEMBL4718043

SCHEMBL4718043

O=CNCCCc1nc2ncccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
HCAR2 Q8TDS4 4/20 0.42
NUDT1 P36639 1/20 0.42
DAGLA Q9Y4D2 1/20 0.40
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 2/20 0.39
DRD4 P21917 1/20 0.39
HTT P42858 1/20 0.39
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
PDE5A O76074 1/20 0.38
HPSE Q9Y251 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718040 0.81 CYP2C9 (0.45) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL4716249 0.79 POLB (0.66) POLBHTT
SCHEMBL4719992 0.77 NUDT1 (0.53) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL8326986 0.77 NOS1 (0.54) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL9570423 0.76 CYP2C9 (0.53) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL246326 0.76 PDE5A (0.53) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL8325044 0.75 DAGLA (0.53) CYP2C9NOS1NOS2HCAR2NUDT1
SCHEMBL9597011 0.73 CYP2C9 (0.53) CYP2C9NOS1NOS2NUDT1DAGLA
SCHEMBL3960231 0.73 CYP2C9 (0.57) CYP2C9NOS1NOS2NUDT1DRD4
SCHEMBL24823966 0.73 NUDT1 (0.45) CYP2C9NOS1NOS2NUDT1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed